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Target
Isoform Beta of cGMP-dependent protein kinase 1 [5-676,G306E]
Ligand
BDBM65501
Substrate
n/a
Meas. Tech.
Microfluidic Mobility-Shift Assay
pH
7±n/a
EC50
370±13 nM
Comments
extracted
Citation
Campbell, JC; Henning, P; Franz, E; Sankaran, B; Herberg, FW; Kim, C Structural Basis of Analog Specificity in PKG I and II. ACS Chem Biol 12:2388-2398 (2017) [PubMed] Article
More Info.:
Target
Name:
Isoform Beta of cGMP-dependent protein kinase 1 [5-676,G306E]
Synonyms:
KGP1_HUMAN | PRKG1 | PRKG1B | PRKGR1A | PRKGR1B | cGMP-dependent protein kinase 1 [5-676,G306E] | hPKG 1 beta (aa 5-676)
Type:
Protein
Mol. Mass.:
76225.72
Organism:
Human
Description:
Q13976-2 (1-351) (G306E)
Residue:
672
Sequence:
RDLQYALQEKIEELRQRDALIDELELELDQKDELIQKLQNELDKYRSVIRPATQQAQKQSASTLQGEPRTKRQAISAEPTAFDIQDLSHVTLPFYPKSPQSKDLIKEAILDNDFMKNLELSQIQEIVDCMYPVEYGKDSCIIKEGDVGSLVYVMEDGKVEVTKEGVKLCTMGPGKVFGELAILYNCTRTATVKTLVNVKLWAIDRQCFQTIMMRTGLIKHTEYMEFLKSVPTFQSLPEEILSKLADVLEETHYENGEYIIRQGARGDTFFIISKGTVNVTREDSPSEDPVFLRTLGKGDWFGEKALQGEDVRTANVIAAEAVTCLVIDRDSFKHLIGGLDDVSNKAYEDAEAKAKYEAEAAFFANLKLSDFNIIDTLGVGGFGRVELVQLKSEESKTFAMKILKKRHIVDTRQQEHIRSEKQIMQGAHSDFIVRLYRTFKDSKYLYMLMEACLGGELWTILRDRGSFEDSTTRFYTACVVEAFAYLHSKGIIYRDLKPENLILDHRGYAKLVDFGFAKKIGFGKKTWTFCGTPEYVAPEIILNKGHDISADYWSLGILMYELLTGSPPFSGPDPMKTYNIILRGIDMIEFPKKIAKNAANLIKKLCRDNPSERLGNLKNGVKDIQKHKWFEGFNWEGLRKGTLTPPIIPSVASPTDTSNFDSFPEDNDEPPP