Reaction Details Report a problem with these data
Target
cGMP-dependent protein kinase 2 [41-418,G232E]
Ligand
BDBM65501
Substrate
n/a
Meas. Tech.
Microfluidic Mobility-Shift Assay
pH
7±n/a
EC50
184±5.0 nM
Comments
extracted
Citation
Campbell, JC; Henning, P; Franz, E; Sankaran, B; Herberg, FW; Kim, C Structural Basis of Analog Specificity in PKG I and II. ACS Chem Biol 12:2388-2398 (2017) [PubMed] Article
More Info.:
Target
Name:
cGMP-dependent protein kinase 2 [41-418,G232E]
Synonyms:
KGP2_HUMAN | PRKG2 | PRKGR2 | hPKG II 41 418 (G232E)
Type:
n/a
Mol. Mass.:
43354.14
Organism:
Human
Description:
Q13237[41-418,G232E]
Residue:
378
Sequence:
DAEIQEREYHLKELREQLSKQTVAIAELTEELQNKCIQLNKLQDVVHMQGGSPLQASPDKVPLEVHRKTSGLVSLHSRRGAKAGVSAEPTTRTYDLNKPPEFSFEKARVRKDSSEKKLITDALNKNQFLKRLDPQQIKDMVECMYGRNYQQGSYIIKQGEPGNHIFVLAEGRLEVFQGEKLLSSIPMWTTFEELAILYNCTRTASVKAITNVKTWALDREVFQNIMRRTAQARDEQYRNFLRSVSLLKNLPEDKLTKIIDCLEVEYYDKGDYIIREGEEGSTFFILAKGKVKVTQSTEGHDQPQLIKTLQKGEYFGEKALISDDVRSANIIAEENDVACLVIDRETFNQTVGTFEELQKYLEGYVANLNRDDEKRHAK