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Target
Zinc finger protein mex-5
Ligand
BDBM52802
Substrate
n/a
Meas. Tech.
Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2
EC50
300000±n/a nM
Citation
 PubChem, PC Fluorescent Polarization Homogeneous Dose Response HTS to Indentify Inhibitors of Mex-5 Binding to TCR-2 PubChem Bioassay (2009)[AID] 
Target
Name:
Zinc finger protein mex-5
Synonyms:
MEX5_CAEEL | RecName: Full=Zinc finger protein mex-5 | mex-5
Type:
Enzyme Catalytic Domain
Mol. Mass.:
52832.78
Organism:
Caenorhabditis elegans
Description:
gi_55976631
Residue:
468
Sequence:
MKAASNSVSSAGGSVSPTTTQPPLPPGQSSHPQIYDQQMQYYFAAAMPNQPMATYAAQNGSSQQYAPAAPYYQDANGQYVQVPANGSMAPQQHMMVSGQPYLYMAQPQQGAQQVMQSGQPQLIYYQQSMAPQAAPMYFHPMQAAPMLPEQMGVMPHTQPAIPPQQQPRQVGVEISSTRTAPLTSSTPLPTSLEYETVQRDNRNRNIQFRYHRVMEHDELPIDEISKITLDNHNDDTMSAEKENHFHEHRGEKFGRRGFPIPETDSQQPPNYKTRLCMMHASGIKPCDMGARCKFAHGLKELRATDAPARYPNNKYKTKLCKNFARGGTGFCPYGLRCEFVHPTDKEFQNIPPYQRMSHDDQDYDQDVIPEDYVVARHQPRFMRTGGRATTPTKVMLKHRNVAGSMMCLSNAGRDLQAGGDYNQPESNEDDLPPHLRRNRRENPPMNKRRTSLSTKWTSEENLGLRGHY
  
Inhibitor
Name:
BDBM52802
Synonyms:
2-[[(1-allyl-4-quinolylidene)amino]methylene]malononitrile | 2-[[(1-prop-2-enyl-4-quinolinylidene)amino]methylidene]propanedinitrile | 2-[[(1-prop-2-enylquinolin-4-ylidene)amino]methylidene]propanedinitrile | 2-{[1-Allyl-1H-quinolin-(4E)-ylideneamino]-methylene}-malononitrile | MLS001030001 | SMR000427184 | cid_910872
Type:
Small organic molecule
Emp. Form.:
C16H12N4
Mol. Mass.:
260.2933
SMILES:
C=CCn1cc\c(=N/C=C(C#N)C#N)c2ccccc12 |(5.75,6.16,;5.75,4.62,;7.08,3.85,;7.08,2.31,;5.75,1.54,;5.75,,;7.08,-.77,;7.08,-2.31,;5.75,-3.08,;5.75,-4.62,;7.08,-5.39,;8.41,-6.16,;4.41,-5.39,;3.08,-6.16,;8.41,,;9.79,-.82,;11.19,-.03,;11.19,1.57,;9.79,2.36,;8.41,1.54,)|
Structure:
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