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Target
Trans-activator protein BZLF1
Ligand
BDBM62409
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62409
Synonyms:
3-[4-[(3-fluorophenyl)carbamoylamino]piperidino]sulfonylbenzoic acid methyl ester | 3-[[4-[[(3-fluoroanilino)-oxomethyl]amino]-1-piperidinyl]sulfonyl]benzoic acid methyl ester | 3-{4-[3-(3-Fluoro-phenyl)-ureido]-piperidine-1-sulfonyl}-benzoic acid methyl ester | MLS000034134 | SMR000006741 | cid_647747 | methyl 3-[4-[(3-fluorophenyl)carbamoylamino]piperidin-1-yl]sulfonylbenzoate
Type:
Small organic molecule
Emp. Form.:
C20H22FN3O5S
Mol. Mass.:
435.469
SMILES:
COC(=O)c1cccc(c1)S(=O)(=O)N1CCC(CC1)NC(=O)Nc1cccc(F)c1
Structure:
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