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Target
Trans-activator protein BZLF1
Ligand
BDBM62421
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62421
Synonyms:
6-(4-methoxyphenyl)-3-methyl-N-piperonyl-imidazo[2,1-b]thiazole-2-carboxamide | MLS000102114 | N-(1,3-benzodioxol-5-ylmethyl)-6-(4-methoxyphenyl)-3-methyl-2-imidazo[2,1-b]thiazolecarboxamide | N-(1,3-benzodioxol-5-ylmethyl)-6-(4-methoxyphenyl)-3-methyl-imidazo[2,1-b][1,3]thiazole-2-carboxamide | N-(1,3-benzodioxol-5-ylmethyl)-6-(4-methoxyphenyl)-3-methylimidazo[2,1-b][1,3]thiazole-2-carboxamide | SMR000018042 | cid_5310148
Type:
Small organic molecule
Emp. Form.:
C22H19N3O4S
Mol. Mass.:
421.469
SMILES:
COc1ccc(cc1)-c1cn2c(C)c(sc2n1)C(=O)NCc1ccc2OCOc2c1
Structure:
Search PDB for entries with ligand similarity: