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Target
Trans-activator protein BZLF1
Ligand
BDBM62422
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62422
Synonyms:
2-[3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-6-oxo-6H-pyridazin-1-yl]-N-(3-ethoxy-phenyl)-acetamide | 2-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-keto-pyridazin-1-yl]-N-m-phenetyl-acetamide | 2-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-oxidanylidene-pyridazin-1-yl]-N-(3-ethoxyphenyl)ethanamide | 2-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-oxo-1-pyridazinyl]-N-(3-ethoxyphenyl)acetamide | 2-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-oxopyridazin-1-yl]-N-(3-ethoxyphenyl)acetamide | MLS000122621 | SMR000120016 | cid_3224511
Type:
Small organic molecule
Emp. Form.:
C22H21N3O5
Mol. Mass.:
407.4192
SMILES:
CCOc1cccc(NC(=O)Cn2nc(ccc2=O)-c2ccc3OCCOc3c2)c1
Structure:
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