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Target
Trans-activator protein BZLF1
Ligand
BDBM62447
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
HHV-4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62447
Synonyms:
4-N-benzyl-6-morpholin-4-yl-2-N-[(3-nitrophenyl)methylideneamino]-1,3,5-triazine-2,4-diamine | 6-(4-morpholinyl)-N2-[(3-nitrophenyl)methylideneamino]-N4-(phenylmethyl)-1,3,5-triazine-2,4-diamine | 6-morpholin-4-yl-N2-[(3-nitrophenyl)methylideneamino]-N4-(phenylmethyl)-1,3,5-triazine-2,4-diamine | Benzyl-{4-morpholin-4-yl-6-[N'-(3-nitro-benzylidene)-hydrazino]-[1,3,5]triazin-2-yl}-amine | MLS000560376 | SMR000174986 | benzyl-[4-morpholino-6-[N'-(3-nitrobenzylidene)hydrazino]-s-triazin-2-yl]amine | cid_3106798
Type:
Small organic molecule
Emp. Form.:
C21H22N8O3
Mol. Mass.:
434.4512
SMILES:
[O-][N+](=O)c1cccc(CN=Nc2nc(NCc3ccccc3)nc(n2)N2CCOCC2)c1 |w:10.10|
Structure:
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