Reaction Details Report a problem with these data
Target
Trans-activator protein BZLF1
Ligand
BDBM62498
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62498
Synonyms:
2-cyclopropyl-5-[4-[4-(3-methoxyphenyl)piperazin-1-yl]sulfonylphenyl]-1,3-oxazole | 2-cyclopropyl-5-[4-[4-(3-methoxyphenyl)piperazino]sulfonylphenyl]oxazole | 2-cyclopropyl-5-[4-[[4-(3-methoxyphenyl)-1-piperazinyl]sulfonyl]phenyl]oxazole | MLS001095642 | SMR000631514 | cid_16027935
Type:
Small organic molecule
Emp. Form.:
C23H25N3O4S
Mol. Mass.:
439.527
SMILES:
COc1cccc(c1)N1CCN(CC1)S(=O)(=O)c1ccc(cc1)-c1cnc(o1)C1CC1
Structure:
Search PDB for entries with ligand similarity: