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Target
X-box-binding protein 1
Ligand
BDBM34245
Substrate
n/a
Meas. Tech.
XBP1 DR counterscreen for CHOP
IC50
500±n/a nM
Citation
 PubChem, PC XBP1 DR counterscreen for CHOP PubChem Bioassay (2011)[AID] 
Target
Name:
X-box-binding protein 1
Synonyms:
TREB5 | XBP1 | XBP1_HUMAN | XBP2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
28704.14
Organism:
Homo sapiens (Human)
Description:
gi_47678753
Residue:
261
Sequence:
MVVVAAAPNPADGTPKVLLLSGQPASAAGAPAGQALPLMVPAQRGASPEAASGGLPQARKRQRLTHLSPEEKALRRKLKNRVAAQTARDRKKARMSELEQQVVDLEEENQKLLLENQLLREKTHGLVVENQELRQRLGMDALVAEEEAEAKGNEVRPVAGSAESAALRLRAPLQQVQAQLSPLQNISPWILAVLTLQIQSLISCWAFWTTWTQSCSSNALPQSLPAWRSSQRSTQKDPVPYQPPFLCQWGRHQPSWKPLMN
  
Inhibitor
Name:
BDBM34245
Synonyms:
2-hydroxy-6-(piperidine-1-carbonyl)benzo[de]isoquinoline-1,3-dione | 2-hydroxy-6-(piperidine-1-carbonyl)benzo[de]isoquinoline-1,3-quinone | 2-hydroxy-6-[oxo(1-piperidinyl)methyl]benzo[de]isoquinoline-1,3-dione | 2-oxidanyl-6-piperidin-1-ylcarbonyl-benzo[de]isoquinoline-1,3-dione | MLS000080235 | SMR000040360 | cid_659314
Type:
Small organic molecule
Emp. Form.:
C18H16N2O4
Mol. Mass.:
324.3306
SMILES:
ON1C(=O)c2cccc3c(ccc(C1=O)c23)C(=O)N1CCCCC1
Structure:
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