Reaction Details Report a problem with these data
Target
Transmembrane domain-containing protein TMIGD3
Ligand
BDBM50259303
Substrate
n/a
Meas. Tech.
ChEMBL_1691284 (CHEMBL4041933)
Ki
52±n/a nM
Citation
Poli, D; Falsini, M; Varano, F; Betti, M; Varani, K; Vincenzi, F; Pugliese, AM; Pedata, F; Dal Ben, D; Thomas, A; Palchetti, I; Bettazzi, F; Catarzi, D; Colotta, V Imidazo[1,2-a]pyrazin-8-amine core for the design of new adenosine receptor antagonists: Structural exploration to target the A Eur J Med Chem 125:611-628 (2017) [PubMed] Article
More Info.:
Target
Name:
Transmembrane domain-containing protein TMIGD3
Synonyms:
TMIG3_HUMAN | TMIGD3 | Transmembrane domain-containing protein TMIGD3
Type:
PROTEIN
Mol. Mass.:
30335.79
Organism:
Human
Description:
ChEMBL_114868
Residue:
266
Sequence:
MEGSPAGPIEQKEARWESSWEEQPDWTLGCLSPESQFRIPGLPGCILSFQLKVCFLPVMWLFILLSLALISDAMVMDEKVKRSFVLDTASAICNYNAHYKNHPKYWCRGYFRDYCNIIAFSPNSTNHVALRDTGNQLIVTMSCLTKEDTGWYWCGIQRDFARDDMDFTELIVTDDKGTLANDFWSGKDLSGNKTRSCKAPKVVRKADRSRTSILIICILITGLGIISVISHLTKRRRSQRNRRVGNTLKPFSRVLTPKEMAPTEQM