Reaction Details Report a problem with these data
Target
Histone deacetylase 11
Ligand
BDBM50252395
Substrate
n/a
Meas. Tech.
ChEBML_1697945
Ki
495±n/a nM
Citation
Sellmer, A; Stangl, H; Beyer, M; Grünstein, E; Leonhardt, M; Pongratz, H; Eichhorn, E; Elz, S; Striegl, B; Jenei-Lanzl, Z; Dove, S; Straub, RH; Krämer, OH; Mahboobi, S Marbostat-100 Defines a New Class of Potent and Selective Antiinflammatory and Antirheumatic Histone Deacetylase 6 Inhibitors. J Med Chem 61:3454-3477 (2018) [PubMed] Article
More Info.:
Target
Name:
Histone deacetylase 11
Synonyms:
HD11 | HDA11_HUMAN | HDAC11 | Human HDAC11
Type:
Chromatin regulator; hydrolase; repressor
Mol. Mass.:
39187.66
Organism:
Human
Description:
Q96DB2
Residue:
347
Sequence:
MLHTTQLYQHVPETRWPIVYSPRYNITFMGLEKLHPFDAGKWGKVINFLKEEKLLSDSMLVEAREASEEDLLVVHTRRYLNELKWSFAVATITEIPPVIFLPNFLVQRKVLRPLRTQTGGTIMAGKLAVERGWAINVGGGFHHCSSDRGGGFCAYADITLAIKFLFERVEGISRATIIDLDAHQGNGHERDFMDDKRVYIMDVYNRHIYPGDRFAKQAIRRKVELEWGTEDDEYLDKVERNIKKSLQEHLPDVVVYNAGTDILEGDRLGGLSISPAGIVKRDELVFRMVRGRRVPILMVTSGGYQKRTARIIADSILNLFGLGLIGPESPSVSAQNSDTPLLPPAVP