Reaction Details Report a problem with these data
Target
Adenosine receptor A1
Ligand
BDBM50078426
Substrate
n/a
Meas. Tech.
ChEMBL_1701165 (CHEMBL4052147)
Ki
0.864000±n/a nM
Citation
Petrelli, R; Scortichini, M; Kachler, S; Boccella, S; Cerchia, C; Torquati, I; Del Bello, F; Salvemini, D; Novellino, E; Luongo, L; Maione, S; Jacobson, KA; Lavecchia, A; Klotz, KN; Cappellacci, L Exploring the Role of N J Med Chem 60:4327-4341 (2017) [PubMed] Article
More Info.:
Target
Name:
Adenosine receptor A1
Synonyms:
A1 adenosine receptor (hA1) | A1AR | AA1R_HUMAN | ADENOSINE A1 | ADORA1 | Adenosine A1 receptor (A1AR) | Adenosine A1-receptor | Adenosine receptor A1 (A1) | Adenosine receptor A1 (hA1) | Adenosine transporter (AdT)
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
36520.92
Organism:
Human
Description:
P30542
Residue:
326
Sequence:
MPPSISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGALVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKMVVTPRRAAVAIAGCWILSFVVGLTPMFGWNNLSAVERAWAANGSMGEPVIKCEFEKVISMEYMVYFNFFVWVLPPLLLMVLIYLEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALILFLFALSWLPLHILNCITLFCPSCHKPSILTYIAIFLTHGNSAMNPIVYAFRIQKFRVTFLKIWNDHFRCQPAPPIDEDLPEERPDD