Reaction Details Report a problem with these data
Target
Adenosine receptor A2b
Ligand
BDBM50455533
Substrate
n/a
Meas. Tech.
ChEMBL_1754702 (CHEMBL4189462)
Ki
1.3±n/a nM
Citation
Köse, M; Gollos, S; Karcz, T; Fiene, A; Heisig, F; Behrenswerth, A; Kie?-Kononowicz, K; Namasivayam, V; Müller, CE Fluorescent-Labeled Selective Adenosine A J Med Chem 61:4301-4316 (2018) [PubMed] Article
More Info.:
Target
Name:
Adenosine receptor A2b
Synonyms:
AA2BR_MOUSE | Adenosine A2b receptor | Adora2b
Type:
PROTEIN
Mol. Mass.:
36130.09
Organism:
Mouse
Description:
ChEMBL_11831
Residue:
332
Sequence:
MQLETQDALYVALELVIAALAVAGNVLVCAAVGASSALQTPTNYFLVSLATADVAVGLFAIPFAITISLGFCTDFHGCLFLACFVLVLTQSSIFSLLAVAVDRYLAIRVPLRYKGLVTGTRARGIIAVLWVLAFGIGLTPFLGWNSKDSATSNCTELGDGIANKSCCPVTCLFENVVPMSYMVYFNFFGCVLPPLLIMLVIYIKIFMVACKQLQRMELMDHSRTTLQREIHAAKSLAMIVGIFALCWLPVHAINCITLFHPALAKDKPKWVMNVAILLSHANSVVNPIVYAYRNRDFRYSFHKIISRYVLCQAETKGGSGQAGAQSTLSLGL