Reaction Details Report a problem with these data
Target
Beta-casein
Ligand
BDBM50470945
Substrate
n/a
Meas. Tech.
ChEMBL_32297 (CHEMBL646244)
Ki
42±n/a nM
Citation
Giardinà, D; Crucianelli, M; Romanelli, R; Leonardi, A; Poggesi, E; Melchiorre, C Synthesis and biological profile of the enantiomers of [4-(4-amino-6,7-dimethoxyquinazolin-2-yl)-cis-octahydroquinoxalin- 1-yl]furan-2-ylmethanone (cyclazosin), a potent competitive alpha 1B- adrenoceptor antagonist. J Med Chem 39:4602-7 (1996) [PubMed] Article
More Info.:
Target
Name:
Beta-casein
Synonyms:
Beta-casein | CASB_RAT | Csn2 | Csnb
Type:
PROTEIN
Mol. Mass.:
25368.99
Organism:
Rattus norvegicus
Description:
ChEMBL_12483
Residue:
231
Sequence:
MKVFILACLVALALAREKDAFTVSSETGSISSEESVEHINEKLQKVKLMGQVQSEDVLQNKFHSGIQSEPQAIPYAQTISCSPIPQNIQPIAQPPVVPTVGPIISPELESFLKAKATVLPKHKQMPFLNSETVLRLFNSQIPSLDLANLHLPQSPAQLQAQIVQAFPQTPAVVSSQPQLSHPQSKSQYLVQQLAPLFQQGMPVQDLLQYLDLLLNPTLQFLATQQLHSTSV