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Target
Similar to alpha-tubulin isoform 1
Ligand
BDBM50101086
Substrate
n/a
Meas. Tech.
ChEMBL_211347 (CHEMBL815040)
IC50
2200±n/a nM
Citation
 Owa, T; Yokoi, A; Yamazaki, K; Yoshimatsu, K; Yamori, T; Nagasu, T Array-based structure and gene expression relationship study of antitumor sulfonamides including N-[2-[(4-hydroxyphenyl)amino]-3-pyridinyl]-4-methoxybenzenesulfonamide and N-(3-chloro-7-indolyl)-1,4-benzenedisulfonamide. J Med Chem 45:4913-22 (2002) [PubMed]  Article 
Target
Name:
Similar to alpha-tubulin isoform 1
Synonyms:
Similar to alpha-tubulin isoform 1
Type:
PROTEIN
Mol. Mass.:
10383.05
Organism:
Bos taurus
Description:
ChEMBL_104716
Residue:
99
Sequence:
CVSASPSTLARLVSRSAMPAGSSTAWNTAFSPMARCQVTKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRSSSTLSSSSQAKKMP
  
Inhibitor
Name:
BDBM50101086
Synonyms:
CHEMBL20684 | E-7010 | N-(2-(4-hydroxyphenylamino)pyridin-3-yl)-4-methoxybenzenesulfonamide | N-[2-(4-Hydroxy-phenylamino)-pyridin-3-yl]-4-methoxy-benzenesulfonamide | N-{2-[(4-hydroxyphenyl)amino]pyridin-3-yl}-4-methoxybenzenesulfonamide
Type:
Small organic molecule
Emp. Form.:
C18H17N3O4S
Mol. Mass.:
371.41
SMILES:
COc1ccc(cc1)S(=O)(=O)Nc1cccnc1Nc1ccc(O)cc1
Structure:
Search PDB for entries with ligand similarity: