Reaction Details
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Target
Trophozoite cysteine proteinase
Ligand
BDBM50486867
Substrate
n/a
Meas. Tech.
ChEMBL_903031 (CHEMBL3063284)
IC50
800±n/a nM
Citation
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More Info.:
Target
Name:
Trophozoite cysteine proteinase
Synonyms:
3.4.22.- | CYSP_PLAFA | TCP | Trophozoite cysteine proteinase
Type:
PROTEIN
Mol. Mass.:
66893.11
Organism:
Plasmodium falciparum
Description:
ChEMBL_106615
Residue:
569
Sequence:
MVAIKEMKELAFARPSLVETLNKKKKFLKKKEKRTFVLSIYAFITFIIFCIGILYFTNKSSAHNNNNNKNEHSLKKEEIELLRVLLEKYKKQKDGILNESSNEEDEEKYTLNSETYNNKNNVSNIKNDSIKSKKEEYINLERILLEKYKKFINENNEENRKELSNILHKLLEINKLILREEKDDKKVYLINDNYDEKGALEIGMNEEMKYKKEDPINNIKYASKFFKFMKEHNKVYKNIDEQMRKFEIFKINYISIKNHNKLNKNAMYKKKVNQFSDYSEEELKEYFKTLLHVPNHMIEKYSKPFENHLKDNILISEFYTNGKRNEKDIFSKVPEILDYREKGIVHEPKDQGLCGSCWAFASVGNIESVFAKKNKNILSFSEQEVVDCSKDNFGCDGGHPFYSFLYVLQNELCLGDEYKYKAKDDMFCLNYRCKRKVSLSSIGAVKENQLILALNEVGPLSVNVGVNNDFVAYSEGVYNGTCSEELNHSVLLVGYGQVEKTKLNYNNKIQTYNTKENSNQPDDNIIYYWIIKNSWSKKWGENGFMRLSRNKNGDNVFCGIGEEVFYPIL