Reaction Details
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Target
Phosphodiesterase
Ligand
BDBM50487528
Substrate
n/a
Meas. Tech.
ChEMBL_909521 (CHEMBL3055687)
IC50
2432000±n/a nM
Citation
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More Info.:
Target
Name:
Phosphodiesterase
Synonyms:
3.1.4.- | PDE7B | Phosphodiesterase
Type:
PROTEIN
Mol. Mass.:
50563.76
Organism:
Bos taurus
Description:
ChEMBL_106550
Residue:
438
Sequence:
MPVLERYFHSAELGRRWTAPEGELPAPLGSRPGCQQGPLPWDLPEMIRMVKLVWKSKSELQATKQRGILENEDALHSIPGDVRLRGQTGVPAERRGSYPFIDFRLLNNTTHSGEIGTKKKVKRLLSFQRYFHASRLLRGIIPQAPLHLLDEDYLGQARHMLSKVGMWDFDIFLFDRLTNGNSLVTLLCHLFNTHGLIHHFKLDMVTLHRFLVMVQEDYHSQNPYHNAVHAADVTQAMHCYLKEPKLASFLTPLDIMLGLLAAAAHDVDHPGVNQPFLIKTNHHLANLYQNMSVLENHHWRSTIGMLRESRLLAHLPKEMTQDIEQQLGSLILATDINRQNEFLTRLKAHLHNKDLRLEEVHDRHFMLQIALKCADICNPCRIWEMSKQWSERVCEEFYRQGDLEQKFELEISPLCNQQKDSIPSIQIGELSSIVILNE