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Target
Potassium channel subfamily K member 5
Ligand
BDBM50123519
Substrate
n/a
Meas. Tech.
ChEMBL_1822389 (CHEMBL4322153)
IC50
12000±n/a nM
Citation
Bedoya, M; Rinné, S; Kiper, AK; Decher, N; González, W; Ramírez, D TASK Channels Pharmacology: New Challenges in Drug Design. J Med Chem 62:10044-10058 (2019) [PubMed] Article
More Info.:
Target
Name:
Potassium channel subfamily K member 5
Synonyms:
Acid-sensitive potassium channel protein TASK-2 | KCNK5 | KCNK5_HUMAN | Potassium channel subfamily K member 5 | TASK2 | TWIK-related acid-sensitive K(+) channel 2
Type:
PROTEIN
Mol. Mass.:
55130.28
Organism:
Human
Description:
ChEMBL_118907
Residue:
499
Sequence:
MVDRGPLLTSAIIFYLAIGAAIFEVLEEPHWKEAKKNYYTQKLHLLKEFPCLGQEGLDKILEVVSDAAGQGVAITGNQTFNNWNWPNAMIFAATVITTIGYGNVAPKTPAGRLFCVFYGLFGVPLCLTWISALGKFFGGRAKRLGQFLTKRGVSLRKAQITCTVIFIVWGVLVHLVIPPFVFMVTEGWNYIEGLYYSFITISTIGFGDFVAGVNPSANYHALYRYFVELWIYLGLAWLSLFVNWKVSMFVEVHKAIKKRRRRRKESFESSPHSRKALQVKGSTASKDVNIFSFLSKKEETYNDLIKQIGKKAMKTSGGGETGPGPGLGPQGGGLPALPPSLVPLVVYSKNRVPTLEEVSQTLRSKGHVSRSPDEEAVARAPEDSSPAPEVFMNQLDRISEECEPWDAQDYHPLIFQDASITFVNTEAGLSDEETSKSSLEDNLAGEESPQQGAEAKAPLNMGEFPSSSESTFTSTESELSVPYEQLMNEYNKANSPKGT