Reaction Details
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Target
Acid-sensing ion channel 1
Ligand
BDBM50510050
Substrate
n/a
Meas. Tech.
ChEMBL_1839999 (CHEMBL4340214)
IC50
>30000±n/a nM
Citation
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More Info.:
Target
Name:
Acid-sensing ion channel 1
Synonyms:
ASIC1_MOUSE | Accn2 | Acid-sensing ion channel | Acid-sensing ion channel 1 | Amiloride-sensitive cation channel 2, neuronal | Asic | Asic1 | Bnac2 | Brain sodium channel 2
Type:
PROTEIN
Mol. Mass.:
59657.36
Organism:
Mus musculus
Description:
ChEMBL_119368
Residue:
526
Sequence:
MELKTEEEEVGGVQPVSIQAFASSSTLHGLAHIFSYERLSLKRALWALCFLGSLAVLLCVCTERVQYYFCYHHVTKLDEVAASQLTFPAVTLCNLNEFRFSQVSKNDLYHAGELLALLNNRYEIPDTQMADEKQLEILQDKANFRSFKPKPFNMREFYDRAGHDIRDMLLSCHFRGEACSAEDFKVVFTRYGKCYTFNSGQDGRPRLKTMKGGTGNGLEIMLDIQQDEYLPVWGETDETSFEAGIKVQIHSQDEPPFIDQLGFGVAPGFQTFVSCQEQRLIYLPSPWGTCNAVTMDSDFFDSYSITACRIDCETRYLVENCNCRMVHMPGDAPYCTPEQYKECADPALDFLVEKDQEYCVCEMPCNLTRYGKELSMVKIPSKASAKYLAKKFNKSEQYIGENILVLDIFFEVLNYETIEQKKAYEIAGLLGDIGGQMGLFIGASILTVLELFDYAYEVIKHRLCRRGKCQKEAKRNSADKGVALSLDDVKRHNPCESLRGHPAGMTYAANILPHHPARGTFEDFTC