Reaction Details Report a problem with these data
Target
Proteasome subunit beta type-5
Ligand
BDBM50516759
Substrate
n/a
Meas. Tech.
ChEMBL_1866705 (CHEMBL4367680)
Ki
17±n/a nM
Citation
Fernandes, GFS; Denny, WA; Dos Santos, JL Boron in drug design: Recent advances in the development of new therapeutic agents. Eur J Med Chem 179:791-804 (2019) [PubMed] Article
More Info.:
Target
Name:
Proteasome subunit beta type-5
Synonyms:
20S proteasome chymotrypsin-like | 26S proteosome | LMPX | MB1 | PSB5_HUMAN | PSMB5 | Proteasome Macropain subunit MB1 | Proteasome subunit beta type-1/beta type-5 | X
Type:
Protein
Mol. Mass.:
28480.96
Organism:
Human
Description:
n/a
Residue:
263
Sequence:
MALASVLERPLPVNQRGFFGLGGRADLLDLGPGSLSDGLSLAAPGWGVPEEPGIEMLHGTTTLAFKFRHGVIVAADSRATAGAYIASQTVKKVIEINPYLLGTMAGGAADCSFWERLLARQCRIYELRNKERISVAAASKLLANMVYQYKGMGLSMGTMICGWDKRGPGLYYVDSEGNRISGATFSVGSGSVYAYGVMDRGYSYDLEVEQAYDLARRAIYQATYRDAYSGGAVNLYHVREDGWIRVSSDNVADLHEKYSGSTP