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Target
Melanin-concentrating hormone receptor 1
Ligand
BDBM50192518
Substrate
n/a
Meas. Tech.
ChEMBL_391843 (CHEMBL861265)
Ki
3.3±n/a nM
Citation
Ma, V; Bannon, AW; Baumgartner, J; Hale, C; Hsieh, F; Hulme, C; Rorrer, K; Salon, J; van Staden, C; Tempest, P Solid-phase synthesis and structure-activity relationships of novel biarylethers as melanin-concentrating hormone receptor-1 antagonists. Bioorg Med Chem Lett 16:5066-72 (2006) [PubMed] Article
More Info.:
Target
Name:
Melanin-concentrating hormone receptor 1
Synonyms:
Gpr24 | MCHR1_MOUSE | Mchr1 | Slc1
Type:
PROTEIN
Mol. Mass.:
39133.74
Organism:
Mouse
Description:
ChEMBL_818502
Residue:
353
Sequence:
MDLQASLLSTGPNASNISDGQDNFTLAGPPPRTRSVSYINIIMPSVFGTICLLGIVGNSTVIFAVVKKSKLHWCSNVPDIFIINLSVVDLLFLLGMPFMIHQLMGNGVWHFGETMCTLITAMDANSQFTSTYILTAMAIDRYLATVHPISSTKFRKPSMATLVICLLWALSFISITPVWLYARLIPFPGGAVGCGIRLPNPDTDLYWFTLYQFFLAFALPFVVITAAYVKILQRMTSSVAPASQRSIRLRTKRVTRTAIAICLVFFVCWAPYYVLQLTQLSISRPTLTFVYLYNAAISLGYANSCLNPFVYIVLCETFRKRLVLSVKPAAQGQLRTVSNAQTADEERTESKGT