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Target
Chymotrypsin-like elastase family member 2A
Ligand
BDBM50281089
Substrate
n/a
Meas. Tech.
ChEMBL_194721 (CHEMBL807702)
IC50
500±n/a nM
Citation
Adonias, M; Anayaba, J; Cámara, J; Canet, E; Gateau-Olesker, A; Gero, SD; Grande, M; Hernando, JI Enantioselective synthesis and antielastase activity of 1,3,4-trisubstituted and 3,4-disubstituted β-lactam antibiotics Bioorg Med Chem Lett 3:2547-2552 (1993) Article
More Info.:
Target
Name:
Chymotrypsin-like elastase family member 2A
Synonyms:
CEL2A_RAT | Cela2a | Ela2 | Ela2a | Elastase 2A | Elastase-2 | Elastase-2A
Type:
PROTEIN
Mol. Mass.:
28894.94
Organism:
Rattus norvegicus
Description:
ChEMBL_194721
Residue:
271
Sequence:
MIRTLLLSALVAGALSCGYPTYEVQHDVSRVVGGQEASPNSWPWQVSLQYLSSGKWHHTCGGSLVANNWVLTAAHCISNSRTYRVLLGRHSLSTSESGSLAVQVSKLVVHEKWNAQKLSNGNDIALVKLASPVALTSKIQTACLPPAGTILPNNYPCYVTGWGRLQTNGATPDVLQQGRLLVVDYATCSSASWWGSSVKTNMVCAGGDGVTSSCNGDSGGPLNCQASNGQWQVHGIVSFGSTLGCNYPRKPSVFTRVSNYIDWINSVIAKN