Reaction Details Report a problem with these data
Target
Cathepsin L2
Ligand
BDBM50336480
Substrate
n/a
Meas. Tech.
ChEMBL_716901 (CHEMBL1670880)
Ki
4200±n/a nM
Citation
Severino, RP; Guido, RV; Marques, EF; Brömme, D; da Silva, MF; Fernandes, JB; Andricopulo, AD; Vieira, PC Acridone alkaloids as potent inhibitors of cathepsin V. Bioorg Med Chem 19:1477-81 (2011) [PubMed] Article
More Info.:
Target
Name:
Cathepsin L2
Synonyms:
CATL2 | CATL2_HUMAN | CTSL2 | CTSU | CTSV | Cathepsin U | Cathepsin V
Type:
Enzyme
Mol. Mass.:
37341.06
Organism:
Human
Description:
O60911
Residue:
334
Sequence:
MNLSLVLAAFCLGIASAVPKFDQNLDTKWYQWKATHRRLYGANEEGWRRAVWEKNMKMIELHNGEYSQGKHGFTMAMNAFGDMTNEEFRQMMGCFRNQKFRKGKVFREPLFLDLPKSVDWRKKGYVTPVKNQKQCGSCWAFSATGALEGQMFRKTGKLVSLSEQNLVDCSRPQGNQGCNGGFMARAFQYVKENGGLDSEESYPYVAVDEICKYRPENSVANDTGFTVVAPGKEKALMKAVATVGPISVAMDAGHSSFQFYKSGIYFEPDCSSKNLDHGVLVVGYGFEGANSNNSKYWLVKNSWGPEWGSNGYVKIAKDKNNHCGIATAASYPNV