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Target
P2Y purinoceptor 1
Ligand
BDBM50409654
Substrate
n/a
Meas. Tech.
ChEMBL_147710 (CHEMBL759180)
EC50
1±n/a nM
Citation
 Nahum, V; Zündorf, G; Lévesque, SA; Beaudoin, AR; Reiser, G; Fischer, B Adenosine 5'-O-(1-boranotriphosphate) derivatives as novel P2Y(1) receptor agonists. J Med Chem 45:5384-96 (2002) [PubMed]  Article 
Target
Name:
P2Y purinoceptor 1
Synonyms:
ATP receptor | P2RY1_RAT | P2Y1 | P2ry1 | Purinergic receptor | Purinergic receptor P2Y1
Type:
PROTEIN
Mol. Mass.:
42338.46
Organism:
Rattus norvegicus
Description:
ChEMBL_873671
Residue:
373
Sequence:
MTEVPWSAVPNGTDAAFLAGLGSLWGNSTIASTAAVSSSFRCALIKTGFQFYYLPAVYILVFIIGFLGNSVAIWMFVFHMKPWSGISVYMFNLALADFLYVLTLPALIFYYFNKTDWIFGDVMCKLQRFIFHVNLYGSILFLTCISAHRYSGVVYPLKSLGRLKKKNAIYVSVLVWLIVVVAISPILFYSGTGIRKNKTVTCYDSTSDEYLRSYFIYSMCTTVAMFCIPLVLILGCYGLIVRALIYKDLDNSPLRRKSIYLVIIVLTVFAVSYIPFHVMKTMNLRARLDFQTPEMCDFNDRVYATYQVTRGLASLNSCVDPILYFLAGDTFRRRLSRATRKASRRSEANLQSKSEEMTLNILSEFKQNGDTSL
  
Inhibitor
Name:
BDBM50409654
Synonyms:
CHEMBL2021421
Type:
Small organic molecule
Emp. Form.:
C10H14BClN5O12P3
Mol. Mass.:
535.432
SMILES:
[BH3-]P(=O)(OC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)nc(Cl)nc12)OP([O-])(=O)OP([O-])([O-])=O |r|
Structure:
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