Reaction Details
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Target
Potassium voltage-gated channel subfamily D member 2
Ligand
BDBM50213092
Substrate
n/a
Meas. Tech.
ChEMBL_436810 (CHEMBL905112)
IC50
17000±n/a nM
Citation
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More Info.:
Target
Name:
Potassium voltage-gated channel subfamily D member 2
Synonyms:
KCND2_RAT | Kcnd2 | RK5 | Shal1 | Voltage-gated potassium channel subunit Kv4.2
Type:
PROTEIN
Mol. Mass.:
70560.86
Organism:
Rattus norvegicus
Description:
ChEMBL_436810
Residue:
630
Sequence:
MAAGVAAWLPFARAAAIGWMPVASGPMPAPPRQERKRTQDALIVLNVSGTRFQTWQDTLERYPDTLLGSSERDFFYHPETQQYFFDRDPDIFRHILNFYRTGKLHYPRHECISAYDEELAFFGLIPEIIGDCCYEEYKDRRRENAERLQDDADTDNTGESALPTMTARQRVWRAFENPHTSTMALVFYYVTGFFIAVSVIANVVETVPCGSSPGHIKELPCGERYAVAFFCLDTACVMIFTVEYLLRLAAAPSRYRFVRSVMSIIDVVAILPYYIGLVMTDNEDVSGAFVTLRVFRVFRIFKFSRHSQGLRILGYTLKSCASELGFLLFSLTMAIIIFATVMFYAEKGSSASKFTSIPAAFWYTIVTMTTLGYGDMVPKTIAGKIFGSICSLSGVLVIALPVPVIVSNFSRIYHQNQRADKRRAQKKARLARIRAAKSGSANAYMQSKRNGLLSNQLQSSEDEPAFVSKSGSSFETQHHHLLHCLEKTTNHEFVDEQVFEESCMEVATVNRPSSHSPSLSSQQGVTSTCCSRRHKKSFRIPNANVSGSHRGSVQELSTIQIRCVERTPLSNSRSSLNAKMEECVKLNCEQPYVTTAIISIPTPPVTTPEGDDRPESPEYSGGNIVRVSAL