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Target
Arginase-1
Ligand
BDBM50375814
Substrate
n/a
Meas. Tech.
ChEMBL_474406 (CHEMBL938291)
Ki
17100±n/a nM
Citation
Kotthaus, J; Schade, D; Töpker-Lehmann, K; Beitz, E; Clement, B N(delta)-Methylated L-arginine derivatives and their effects on the nitric oxide generating system. Bioorg Med Chem 16:2305-12 (2008) [PubMed] Article
More Info.:
Target
Name:
Arginase-1
Synonyms:
ARG1 | ARGI1_BOVIN | Liver-type arginase | Type I arginase
Type:
PROTEIN
Mol. Mass.:
35008.90
Organism:
Bos taurus
Description:
ChEMBL_474406
Residue:
322
Sequence:
MSSKPQSIGVIGAPFSKGQPRGGVEEGPTVLRKAGLLEKLKELECDVKDYGDLSFADNLDDSPFQIVKNPRCVGKASEKLADVVAEVKKTGRISLVLGGDHSLAIGSISGHARVHPDLCVIWVDAHTDINTPLTTKTGNLHGQPVSFLLKELKEKMPEVPGFYWVAPCISAKDIVYIGLRDVDPGEHYILKTLGIKYFSMTEVDKLGIGKVMEETFSYLLGRKKRPIHLSFDVDGLDPSFTPATGTPVQGGLTYREGLYITEEIYKTGLLSGLDIMEVNPSLGKTPEEVTRTVNTTVAITMACFGVAREGNHKPIDYLSPPK