Reaction Details Report a problem with these data
Target
Adenosine receptor A3
Ligand
BDBM50395122
Substrate
n/a
Meas. Tech.
ChEMBL_859652 (CHEMBL2168889)
Ki
450±n/a nM
Citation
Korboukh, I; Hull-Ryde, EA; Rittiner, JE; Randhawa, AS; Coleman, J; Fitzpatrick, BJ; Setola, V; Janzen, WP; Frye, SV; Zylka, MJ; Jin, J Orally active adenosine A(1) receptor agonists with antinociceptive effects in mice. J Med Chem 55:6467-77 (2012) [PubMed] Article
More Info.:
Target
Name:
Adenosine receptor A3
Synonyms:
A3 adenosine receptor (hA3) | AA3R_HUMAN | ADORA3 | Adenosine A3 receptor (A3AR)
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
36197.32
Organism:
Human
Description:
P0DMS8
Residue:
318
Sequence:
MPNNSTALSLANVTYITMEIFIGLCAIVGNVLVICVVKLNPSLQTTTFYFIVSLALADIAVGVLVMPLAIVVSLGITIHFYSCLFMTCLLLIFTHASIMSLLAIAVDRYLRVKLTVRYKRVTTHRRIWLALGLCWLVSFLVGLTPMFGWNMKLTSEYHRNVTFLSCQFVSVMRMDYMVYFSFLTWIFIPLVVMCAIYLDIFYIIRNKLSLNLSNSKETGAFYGREFKTAKSLFLVLFLFALSWLPLSIINCIIYFNGEVPQLVLYMGILLSHANSMMNPIVYAYKIKKFKETYLLILKACVVCHPSDSLDTSIEKNSE