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Target
Dual specificity protein phosphatase 23
Ligand
BDBM50436357
Substrate
n/a
Meas. Tech.
ChEMBL_966891 (CHEMBL2401182)
IC50
5700±n/a nM
Citation
He, Y; Liu, S; Menon, A; Stanford, S; Oppong, E; Gunawan, AM; Wu, L; Wu, DJ; Barrios, AM; Bottini, N; Cato, AC; Zhang, ZY A potent and selective small-molecule inhibitor for the lymphoid-specific tyrosine phosphatase (LYP), a target associated with autoimmune diseases. J Med Chem 56:4990-5008 (2013) [PubMed] Article
More Info.:
Target
Name:
Dual specificity protein phosphatase 23
Synonyms:
DUS23_HUMAN | DUSP23 | Dual specificity protein phosphatase 23 | Dual specificity protein phosphatase 23 (VHZ) | LDP-3 | LDP3 | Low molecular mass dual specificity phosphatase 3 | VH1-like phosphatase Z | VHZ
Type:
Enzyme
Mol. Mass.:
16592.49
Organism:
Homo sapiens (Human)
Description:
Q9BVJ7
Residue:
150
Sequence:
MGVQPPNFSWVLPGRLAGLALPRLPAHYQFLLDLGVRHLVSLTERGPPHSDSCPGLTLHRLRIPDFCPPAPDQIDRFVQIVDEANARGEAVGVHCALGFGRTGTMLACYLVKERGLAAGDAIAEIRRLRPGSIETYEQEKAVFQFYQRTK