Reaction Details Report a problem with these data
Target
Somatostatin receptor type 3
Ligand
BDBM50021064
Substrate
n/a
Meas. Tech.
ChEMBL_1365873 (CHEMBL3296531)
Ki
6.8±n/a nM
Citation
Li, D; Wu, Z; Yu, Y; Ball, RG; Guo, L; Sherer, E; He, S; Hong, Q; Lai, Z; Qi, H; Truong, Q; Yang, DX; Chicchi, GG; Tsao, KL; Trusca, D; Trujillo, M; Pachanski, M; Eiermann, GJ; Howard, AD; Zhou, YP; Zhang, BB; Nargund, RP; Hagmann, WK Diamine Derivatives as Novel Small-Molecule, Potent, and Subtype-Selective Somatostatin SST3 Receptor Agonists. ACS Med Chem Lett 5:690-5 (2014) [PubMed] Article
More Info.:
Target
Name:
Somatostatin receptor type 3
Synonyms:
SOMATOSTATIN SST3 | SS-3-R | SS3-R | SS3R | SSR-28 | SSR3_HUMAN | SSTR3 | Somatostatin receptor type 3 (SSTR3)
Type:
Protein
Mol. Mass.:
45855.97
Organism:
Human
Description:
P32745
Residue:
418
Sequence:
MDMLHPSSVSTTSEPENASSAWPPDATLGNVSAGPSPAGLAVSGVLIPLVYLVVCVVGLLGNSLVIYVVLRHTASPSVTNVYILNLALADELFMLGLPFLAAQNALSYWPFGSLMCRLVMAVDGINQFTSIFCLTVMSVDRYLAVVHPTRSARWRTAPVARTVSAAVWVASAVVVLPVVVFSGVPRGMSTCHMQWPEPAAAWRAGFIIYTAALGFFGPLLVICLCYLLIVVKVRSAGRRVWAPSCQRRRRSERRVTRMVVAVVALFVLCWMPFYVLNIVNVVCPLPEEPAFFGLYFLVVALPYANSCANPILYGFLSYRFKQGFRRVLLRPSRRVRSQEPTVGPPEKTEEEDEEEEDGEESREGGKGKEMNGRVSQITQPGTSGQERPPSRVASKEQQLLPQEASTGEKSSTMRISYL