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Target
Probable G-protein coupled receptor 34
Ligand
BDBM50096438
Substrate
n/a
Meas. Tech.
ChEMBL_1495908 (CHEMBL3579719)
EC50
>1000±n/a nM
Citation
Ikubo, M; Inoue, A; Nakamura, S; Jung, S; Sayama, M; Otani, Y; Uwamizu, A; Suzuki, K; Kishi, T; Shuto, A; Ishiguro, J; Okudaira, M; Kano, K; Makide, K; Aoki, J; Ohwada, T Structure-activity relationships of lysophosphatidylserine analogs as agonists of G-protein-coupled receptors GPR34, P2Y10, and GPR174. J Med Chem 58:4204-19 (2015) [PubMed] Article
More Info.:
Target
Name:
Probable G-protein coupled receptor 34
Synonyms:
GPR34 | GPR34_HUMAN | Probable G-protein coupled receptor 34
Type:
PROTEIN
Mol. Mass.:
43892.32
Organism:
Human
Description:
ChEMBL_109761
Residue:
381
Sequence:
MRSHTITMTTTSVSSWPYSSHRMRFITNHSDQPPQNFSATPNVTTCPMDEKLLSTVLTTSYSVIFIVGLVGNIIALYVFLGIHRKRNSIQIYLLNVAIADLLLIFCLPFRIMYHINQNKWTLGVILCKVVGTLFYMNMYISIILLGFISLDRYIKINRSIQQRKAITTKQSIYVCCIVWMLALGGFLTMIILTLKKGGHNSTMCFHYRDKHNAKGEAIFNFILVVMFWLIFLLIILSYIKIGKNLLRISKRRSKFPNSGKYATTARNSFIVLIIFTICFVPYHAFRFIYISSQLNVSSCYWKEIVHKTNEIMLVLSSFNSCLDPVMYFLMSSNIRKIMCQLLFRRFQGEPSRSESTSEFKPGYSLHDTSVAVKIQSSSKST