Reaction Details Report a problem with these data
Target
Carbonic anhydrase
Ligand
BDBM26985
Substrate
n/a
Meas. Tech.
ChEMBL_1504763 (CHEMBL3595048)
Ki
5800000±n/a nM
Citation
De Luca, V; Vullo, D; Del Prete, S; Carginale, V; Scozzafava, A; Osman, SM; AlOthman, Z; Supuran, CT; Capasso, C Cloning, characterization and anion inhibition studies of a new¿-carbonic anhydrase from the Antarctic bacterium Pseudoalteromonas haloplanktis. Bioorg Med Chem 23:4405-9 (2015) [PubMed] Article
More Info.:
Target
Name:
Carbonic anhydrase
Synonyms:
CAH_METTT | CAM | Carbonic anhydrase | Gamma-carbonic anhydrase
Type:
Protein
Mol. Mass.:
26390.56
Organism:
Methanosarcina thermophila
Description:
P40881
Residue:
247
Sequence:
MMFNKQIFTILILSLSLALAGSGCISEGAEDNVAQEITVDEFSNIRENPVTPWNPEPSAPVIDPTAYIDPQASVIGEVTIGANVMVSPMASIRSDEGMPIFVGDRSNVQDGVVLHALETINEEGEPIEDNIVEVDGKEYAVYIGNNVSLAHQSQVHGPAAVGDDTFIGMQAFVFKSKVGNNCVLEPRSAAIGVTIPDGRYIPAGMVVTSQAEADKLPEVTDDYAYSHTNEAVVYVNVHLAEGYKETS