Reaction Details
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Target
Rhodopsin kinase GRK7
Ligand
BDBM50135286
Substrate
n/a
Meas. Tech.
ChEMBL_1546680 (CHEMBL3748205)
IC50
>10000±n/a nM
Citation
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More Info.:
Target
Name:
Rhodopsin kinase GRK7
Synonyms:
G protein-coupled receptor kinase 7 | GPRK7 | GRK7 | GRK7_HUMAN
Type:
PROTEIN
Mol. Mass.:
62210.84
Organism:
Homo sapiens (Human)
Description:
ChEMBL_774199
Residue:
553
Sequence:
MVDMGALDNLIANTAYLQARKPSDCDSKELQRRRRSLALPGLQGCAELRQKLSLNFHSLCEQQPIGRRLFRDFLATVPTFRKAATFLEDVQNWELAEEGPTKDSALQGLVATCASAPAPGNPQPFLSQAVATKCQAATTEEERVAAVTLAKAEAMAFLQEQPFKDFVTSAFYDKFLQWKLFEMQPVSDKYFTEFRVLGKGGFGEVCAVQVKNTGKMYACKKLDKKRLKKKGGEKMALLEKEILEKVSSPFIVSLAYAFESKTHLCLVMSLMNGGDLKFHIYNVGTRGLDMSRVIFYSAQIACGMLHLHELGIVYRDMKPENVLLDDLGNCRLSDLGLAVEMKGGKPITQRAGTNGYMAPEILMEKVSYSYPVDWFAMGCSIYEMVAGRTPFKDYKEKVSKEDLKQRTLQDEVKFQHDNFTEEAKDICRLFLAKKPEQRLGSREKSDDPRKHHFFKTINFPRLEAGLIEPPFVPDPSVVYAKDIAEIDDFSEVRGVEFDDKDKQFFKNFATGAVPIAWQEEIIETGLFEELNDPNRPTGCEEGNSSKSGVCLLL