Reaction Details
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Target
Activin receptor type-2B
Ligand
BDBM50183449
Substrate
n/a
Meas. Tech.
ChEMBL_1586819 (CHEMBL3826651)
IC50
7680±n/a nM
Citation
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More Info.:
Target
Name:
Activin receptor type-2B
Synonyms:
ACVR2B | AVR2B_HUMAN | Activin receptor type-2B
Type:
Enzyme Catalytic Domain
Mol. Mass.:
57713.76
Organism:
Homo sapiens (Human)
Description:
gi_116734708
Residue:
512
Sequence:
MTAPWVALALLWGSLCAGSGRGEAETRECIYYNANWELERTNQSGLERCEGEQDKRLHCYASWRNSSGTIELVKKGCWLDDFNCYDRQECVATEENPQVYFCCCEGNFCNERFTHLPEAGGPEVTYEPPPTAPTLLTVLAYSLLPIGGLSLIVLLAFWMYRHRKPPYGHVDIHEDPGPPPPSPLVGLKPLQLLEIKARGRFGCVWKAQLMNDFVAVKIFPLQDKQSWQSEREIFSTPGMKHENLLQFIAAEKRGSNLEVELWLITAFHDKGSLTDYLKGNIITWNELCHVAETMSRGLSYLHEDVPWCRGEGHKPSIAHRDFKSKNVLLKSDLTAVLADFGLAVRFEPGKPPGDTHGQVGTRRYMAPEVLEGAINFQRDAFLRIDMYAMGLVLWELVSRCKAADGPVDEYMLPFEEEIGQHPSLEELQEVVVHKKMRPTIKDHWLKHPGLAQLCVTIEECWDHDAEARLSAGCVEERVSLIRRSVNGTTSDCLVSLVTSVTNVDLPPKESSI