Reaction Details Report a problem with these data
Target
Galanin receptor type 3
Ligand
BDBM97192
Substrate
n/a
IC50
391.72±n/a nM
Citation
 PubChem, PC Fluorescence-based cell-based primary high throughput dose response assay to identify antagonists of the Galanin Receptor 3 (GalR3). PubChem Bioassay (2013)[AID] 
Target
Name:
Galanin receptor type 3
Synonyms:
GALNR3 | GALR3 | GALR3_HUMAN | Galanin R3 | Galanin receptor 3 | Galanin receptor type 3
Type:
Enzyme Catalytic Domain
Mol. Mass.:
39599.97
Organism:
Human
Description:
Galanin R3 GALR3 HUMAN::O60755
Residue:
368
Sequence:
MADAQNISLDSPGSVGAVAVPVVFALIFLLGTVGNGLVLAVLLQPGPSAWQEPGSTTDLFILNLAVADLCFILCCVPFQATIYTLDAWLFGALVCKAVHLLIYLTMYASSFTLAAVSVDRYLAVRHPLRSRALRTPRNARAAVGLVWLLAALFSAPYLSYYGTVRYGALELCVPAWEDARRRALDVATFAAGYLLPVAVVSLAYGRTLRFLWAAVGPAGAAAAEARRRATGRAGRAMLAVAALYALCWGPHHALILCFWYGRFAFSPATYACRLASHCLAYANSCLNPLVYALASRHFRARFRRLWPCGRRRRHRARRALRRVRPASSGPPGCPGDARPSGRLLAGGGQGPEPREGPVHGGEAARGPE
  
Inhibitor
Name:
BDBM97192
Synonyms:
2-amino-N-(4-phenylbenzyl)quinoline-3-carboxamide | 2-amino-N-(biphenyl-4-ylmethyl)quinoline-3-carboxamide | 2-amino-N-[(4-phenylphenyl)methyl]-3-quinolinecarboxamide | 2-amino-N-[(4-phenylphenyl)methyl]quinoline-3-carboxamide | 2-azanyl-N-[(4-phenylphenyl)methyl]quinoline-3-carboxamide | MLS003678910 | SMR002356458 | cid_53382850
Type:
Small organic molecule
Emp. Form.:
C23H19N3O
Mol. Mass.:
353.4165
SMILES:
Nc1nc2ccccc2cc1C(=O)NCc1ccc(cc1)-c1ccccc1
Structure:
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