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Target
Tyrosine-protein kinase SYK [2-635]
Ligand
BDBM222934
Substrate
n/a
Meas. Tech.
Chip Based Microfluidic Mobility Shift Assay
pH
7.5±n/a
Temperature
303.15±n/a K
IC50
1.3±n/a nM
Comments
extracted
Citation
Buehlmayer, P; Smith, AB; Thoma, G; Van Eis, M Bicyclic heteroaryl cycloalkyldiamine derivatives US Patent US9315500 Publication Date 4/19/2016
More Info.:
Target
Name:
Tyrosine-protein kinase SYK [2-635]
Synonyms:
KSYK_HUMAN | SYK | Tyrosine-protein kinase SYK | Tyrosine-protein kinase SYK (SYK)
Type:
Protein
Mol. Mass.:
71948.80
Organism:
Human
Description:
Human Syk (2-635 aa) (UniProtKB: P43405)
Residue:
634
Sequence:
ASSGMADSANHLPFFFGNITREEAEDYLVQGGMSDGLYLLRQSRNYLGGFALSVAHGRKAHHYTIERELNGTYAIAGGRTHASPADLCHYHSQESDGLVCLLKKPFNRPQGVQPKTGPFEDLKENLIREYVKQTWNLQGQALEQAIISQKPQLEKLIATTAHEKMPWFHGKISREESEQIVLIGSKTNGKFLIRARDNNGSYALCLLHEGKVLHYRIDKDKTGKLSIPEGKKFDTLWQLVEHYSYKADGLLRVLTVPCQKIGTQGNVNFGGRPQLPGSHPATWSAGGIISRIKSYSFPKPGHRKSSPAQGNRQESTVSFNPYEPELAPWAADKGPQREALPMDTEVYESPYADPEEIRPKEVYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNEANDPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVN