Reaction Details Report a problem with these data
Target
chymase
Ligand
BDBM255956
Substrate
n/a
Meas. Tech.
Enzymatic Chymase Assay
pH
7.5±n/a
IC50
2±n/a nM
Comments
extracted
Citation
Fürstner, C; Ackerstaff, J; Straub, A; Meier, H; Tinel, H; Zimmermann, K; Tersteegen, A; Zubov, D; Kast, R; Schamberger, J; Schäfer, M; Börngen, K Bicyclically substituted uracils and the use thereof US Patent US9481672 Publication Date 11/1/2016
More Info.:
Target
Name:
chymase
Synonyms:
n/a
Type:
Enzyme
Mol. Mass.:
27507.42
Organism:
Golden hamster
Description:
A0A1U7QTH6
Residue:
247
Sequence:
MLLPALRLLLFLLGSSAEAGKIIGGTECRPHARPYMAYLEIVTPENHLSACSGFLIRRNFVMTAAHCAGRSITVLLGAHNKKVKEDTWQKLEVEKQFPHPKYDDHLVLNDIMLLKLKEKANLTLGVGTLPISAKSNSIPPGRVCRAVGWGRTNVNEPPSDTLQEVKMRILDPQACKHFEDFHQEPQLCVGNPKKIRNVYKGDSGGPLLCAGIAQGIASYVLRNAKPPSVFTRISHYRPWINKILREN