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Target
Protein-lysine 6-oxidase
Ligand
BDBM469066
Substrate
n/a
Meas. Tech.
LOX Enzyme Activity Assay
IC50
1500±n/a nM
Citation
Springer, C; Marais, R; Niculescu-Duvaz, D; Leung, L; Smithen, D; Callens, C; Tang, H Methylamine derivatives as lysysl oxidase inhibitors for the treatment of cancer US Patent US10807974 Publication Date 10/20/2020
More Info.:
Target
Name:
Protein-lysine 6-oxidase
Synonyms:
LOX | LYOX_PIG
Type:
PROTEIN
Mol. Mass.:
28737.77
Organism:
Sus scrofa
Description:
ChEMBL_108023
Residue:
246
Sequence:
DDPYNPYKYSDDNPYYNYYERPRPGSRYRPGYGTGYFQYGLPDLVPDPYYIQASTYVQKMSMYNLRCAAEENCLASTAYRADVRDYDHRVLLRFPQRVKNQGTSDFLPSRPRYSWEWHSCHQHYHSMDEFSHYDLLDASTQRRVAEGHKASFCLEDTSCDYGYHRRFACTAHTQGLSPGCYDTYNADIDCQWIDITDVKPGNYILKVSVNPSYLVPESDYSNNVVRCEIRYTGHHAYASGCTISPY