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Target
Plasma serine protease inhibitor
Ligand
BDBM528127
Substrate
n/a
Meas. Tech.
Determination of Enzyme Selectivity
IC50
12010±n/a nM
Citation
Davie, RL; Edwards, HJ; Evans, DM; Hodgson, ST; Pethen, SJ; Rooker, DP Pyrazole derivatives as plasma kallikrein inhibitors US Patent US11180484 Publication Date 11/23/2021
More Info.:
Target
Name:
Plasma serine protease inhibitor
Synonyms:
Acrosomal serine protease inhibitor | IPSP_HUMAN | PAI-3 | PAI3 | PCI | PLANH3 | PROCI | Plasminogen activator inhibitor 3 | Protein C inhibitor | SERPINA5 | Serpin A5
Type:
Protein
Mol. Mass.:
45687.25
Organism:
Human
Description:
P05154
Residue:
406
Sequence:
MQLFLLLCLVLLSPQGASLHRHHPREMKKRVEDLHVGATVAPSSRRDFTFDLYRALASAAPSQSIFFSPVSISMSLAMLSLGAGSSTKMQILEGLGLNLQKSSEKELHRGFQQLLQELNQPRDGFQLSLGNALFTDLVVDLQDTFVSAMKTLYLADTFPTNFRDSAGAMKQINDYVAKQTKGKIVDLLKNLDSNAVVIMVNYIFFKAKWETSFNHKGTQEQDFYVTSETVVRVPMMSREDQYHYLLDRNLSCRVVGVPYQGNATALFILPSEGKMQQVENGLSEKTLRKWLKMFKKRQLELYLPKFSIEGSYQLEKVLPSLGISNVFTSHADLSGISNHSNIQVSEMVHKAVVEVDESGTRAAAATGTIFTFRSARLNSQRLVFNRPFLMFIVDNNILFLGKVNRP