Reaction Details
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Target
PEX5-related protein/Peroxisomal membrane protein PEX14
Ligand
BDBM304023
Substrate
n/a
Meas. Tech.
Antitrypanosomal Activity Assay
IC50
15600±n/a nM
Citation
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More Info.:
Target
Name:
PEX5-related protein/Peroxisomal membrane protein PEX14
Synonyms:
PEX14-PEX5
Type:
Enzyme
Mol. Mass.:
n/a
Description:
n/a
Components:
This complex has 2 components.
Component 1
Name:
Peroxisomal membrane protein PEX14
Synonyms:
PEX14 | PEX14_HUMAN | PTS1 receptor-docking protein | Peroxin-14 | Peroxisomal membrane anchor protein PEX14
Type:
Enzyme Catalytic Domain
Mol. Mass.:
41218.98
Organism:
Homo sapiens (Human)
Description:
O75381
Residue:
377
Sequence:
MASSEQAEQPSQPSSTPGSENVLPREPLIATAVKFLQNSRVRQSPLATRRAFLKKKGLTDEEIDMAFQQSGTAADEPSSLGPATQVVPVQPPHLISQPYSPAGSRWRDYGALAIIMAGIAFGFHQLYKKYLLPLILGGREDRKQLERMEAGLSELSGSVAQTVTQLQTTLASVQELLIQQQQKIQELAHELAAAKATTSTNWILESQNINELKSEINSLKGLLLNRRQFPPSPSAPKIPSWQIPVKSPSPSSPAAVNHHSSSDISPVSNESTSSSPGKEGHSPEGSTVTYHLLGPQEEGEGVVDVKGQVRMEVQGEEEKREDKEDEEDEEDDDVSHVDEEDCLGVQREDRRGGDGQINEQVEKLRRPEGASNESERD
Component 2
Name:
PEX5-related protein
Synonyms:
PEX2-related protein | PEX5-like protein | PEX5L | PEX5R | PEX5R_HUMAN | PXR2 | Peroxin-5-related protein | Peroxisome biogenesis factor 5-like | Pex5Rp | TRIP8b | Tetratricopeptide repeat-containing Rab8b-interacting protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
69680.62
Organism:
Homo sapiens (Human)
Description:
Q8IYB4
Residue:
626
Sequence:
MYQGHMQKSKEQGYGKLSSDEDLEIIVDQKQGKGSRAADKAVAMVMKEIPREESAEEKPLLTMTSQLVNEQQESRPLLSPSIDDFLCETKSEAIARPVTSNTAVLTTGLDLLDLSEPVSQTQTKAKKSEPSSKTSSLKKKADGSDLISTDAEQRGQPLRVPETSSLDLDIQTQLEKWDDVKFHGDRNTKGHPMAERKSSSSRTGSKELLWSSEHRSQPELSGGKSALNSESASELELVAPTQARLTKEHRWGSALLSRNHSLEEEFERAKAAVESDTEFWDKMQAEWEEMARRNWISENQEAQNQVTISASEKGYYFHTENPFKDWPGAFEEGLKRLKEGDLPVTILFMEAAILQDPGDAEAWQFLGITQAENENEQAAIVALQRCLELQPNNLKALMALAVSYTNTGHQQDACDALKNWIKQNPKYKYLVKSKKGSPGLTRRMSKSPVDSSVLEGVKELYLEAAHQNGDMIDPDLQTGLGVLFHLSGEFNRAIDAFNAALTVRPEDYSLWNRLGATLANGDRSEEAVEAYTRALEIQPGFIRSRYNLGISCINLGAYREAVSNFLTALSLQRKSRNQQQVPHPAISGNIWAALRIALSLMDQPELFQAANLGDLDVLLRAFNLDP