Reaction Details
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Target
Nuclear receptor ROR-gamma [238-497]
Ligand
BDBM175902
Substrate
n/a
Meas. Tech.
TR-FRET Assay
pH
6.8±n/a
IC50
500±n/a nM
Comments
extracted
Citation
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More Info.:
Target
Name:
Nuclear receptor ROR-gamma [238-497]
Synonyms:
NR1F3 | RORC | RORG | RORG_HUMAN | RZRG | Retinoid-related orphan receptor gamma (RORgamma-LBD)
Type:
Protein
Mol. Mass.:
29835.99
Organism:
Homo sapiens (Human)
Description:
Human RORgamma ligand-binding domain.
Residue:
260
Sequence:
HPGLGELGQGPDSYGSPSFRSTPEAPYASLTEIEHLVQSVCKSYRETCQLRLEDLLRQRSNIFSREEVTGYQRKSMWEMWERCAHHLTEAIQYVVEFAKRLSGFMELCQNDQIVLLKAGAMEVVLVRMCRAYNADNRTVFFEGKYGGMELFRALGCSELISSIFDFSHSLSALHFSEDEIALYTALVLINAHRPGLQEKRKVEQLQYNLELAFHHHLCKTHRQSILAKLPPKGKLRSLCSQHVERLQIFQHLHPIVVQAA