Reaction Details Report a problem with these data
Target
Androgen receptor [633-919]
Ligand
BDBM50529647
Substrate
n/a
Meas. Tech.
Human Androgen Receptor (hAR) Ligand Binding Domain (LBD) Affinity Assay
Ki
28.4±n/a nM
Citation
Narayanan, R; Miller, DD; Ponnusamy, T; Hwang, D; He, Y Selective androgen receptor degrader (SARD) ligands and methods of use US Patent US11648234 Publication Date 5/16/2023
More Info.:
Target
Name:
Androgen receptor [633-919]
Synonyms:
ANDR_HUMAN | AR | Androgen receptor (633-919) | DHTR | NR3C4
Type:
aa 633-919
Mol. Mass.:
33165.80
Organism:
Human
Description:
P10275[633-919]
Residue:
287
Sequence:
KKLGNLKLQEEGEASSTTSPTEETTQKLTVSHIEGYECQPIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHT