Reaction Details Report a problem with these data
Target
Transcriptional enhancer factor TEF-4/Isoform 5 of Transcriptional coactivator [50-100]
Ligand
BDBM626326
Substrate
n/a
Meas. Tech.
HTRF Assay
EC50
130±n/a nM
Citation
Zbieg, JR; Beroza, PP Therapeutic compounds and methods of use US Patent US11787775 Publication Date 10/17/2023
More Info.:
Target
Name:
Transcriptional enhancer factor TEF-4/Isoform 5 of Transcriptional coactivator [50-100]
Synonyms:
TEAD2 YAP50-100 combined
Type:
Protein
Mol. Mass.:
n/a
Description:
n/a
Components:
This complex has 2 components.
Component 1
Name:
Transcriptional enhancer factor TEF-4
Synonyms:
TEA domain family member 2 | TEAD-2 | TEAD2 | TEAD2_HUMAN | TEF4 | Transcriptional enhancer factor TEF-4
Type:
PROTEIN
Mol. Mass.:
49241.42
Organism:
Human
Description:
ChEMBL_119051
Residue:
447
Sequence:
MGEPRAGAALDDGSGWTGSEEGSEEGTGGSEGAGGDGGPDAEGVWSPDIEQSFQEALAIYPPCGRRKIILSDEGKMYGRNELIARYIKLRTGKTRTRKQVSSHIQVLARRKSREIQSKLKDQVSKDKAFQTMATMSSAQLISAPSLQAKLGPTGPQASELFQFWSGGSGPPWNVPDVKPFSQTPFTLSLTPPSTDLPGYEPPQALSPLPPPTPSPPAWQARGLGTARLQLVEFSAFVEPPDAVDSYQRHLFVHISQHCPSPGAPPLESVDVRQIYDKFPEKKGGLRELYDRGPPHAFFLVKFWADLNWGPSGEEAGAGGSISSGGFYGVSSQYESLEHMTLTCSSKVCSFGKQVVEKVETERAQLEDGRFVYRLLRSPMCEYLVNFLHKLRQLPERYMMNSVLENFTILQVVTNRDTQELLLCTAYVFEVSTSERGAQHHIYRLVRD
Component 2
Name:
Isoform 5 of Transcriptional coactivator [50-100]
Synonyms:
Transcriptional coactivator YAP1 (50-100) | YAP1_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
5701.47
Organism:
Human
Description:
P46937-5[50-100]
Residue:
51
Sequence:
AGHQIVHVRGDSETDLEALFNAVMNPKTANVPQTVPMRLRKLPDSFFKPPE