Reaction Details Report a problem with these data
Target
Glycogen [starch] synthase, liver
Ligand
BDBM635135
Substrate
n/a
Meas. Tech.
The GYS2 coupled enzyme assay
IC50
>91760±n/a nM
Citation
Morgans, Jr., DJ; Mellem, K; Powers, HL; Lee, PS; Won, W; Sinz, CJ Inhibitors of glycogen synthase 1 (GYS1) and methods of use thereof US Patent US11814367 Publication Date 11/14/2023
More Info.:
Target
Name:
Glycogen [starch] synthase, liver
Synonyms:
2.4.1.11 | GYS2 | GYS2_HUMAN | Glycogen [starch] synthase, liver
Type:
PROTEIN
Mol. Mass.:
80993.15
Organism:
Human
Description:
ChEMBL_118993
Residue:
703
Sequence:
MLRGRSLSVTSLGGLPQWEVEELPVEELLLFEVAWEVTNKVGGIYTVIQTKAKTTADEWGENYFLIGPYFEHNMKTQVEQCEPVNDAVRRAVDAMNKHGCQVHFGRWLIEGSPYVVLFDIGYSAWNLDRWKGDLWEACSVGIPYHDREANDMLIFGSLTAWFLKEVTDHADGKYVVAQFHEWQAGIGLILSRARKLPIATIFTTHATLLGRYLCAANIDFYNHLDKFNIDKEAGERQIYHRYCMERASVHCAHVFTTVSEITAIEAEHMLKRKPDVVTPNGLNVKKFSAVHEFQNLHAMYKARIQDFVRGHFYGHLDFDLEKTLFLFIAGRYEFSNKGADIFLESLSRLNFLLRMHKSDITVMVFFIMPAKTNNFNVETLKGQAVRKQLWDVAHSVKEKFGKKLYDALLRGEIPDLNDILDRDDLTIMKRAIFSTQRQSLPPVTTHNMIDDSTDPILSTIRRIGLFNNRTDRVKVILHPEFLSSTSPLLPMDYEEFVRGCHLGVFPSYYEPWGYTPAECTVMGIPSVTTNLSGFGCFMQEHVADPTAYGIYIVDRRFRSPDDSCNQLTKFLYGFCKQSRRQRIIQRNRTERLSDLLDWRYLGRYYQHARHLTLSRAFPDKFHVELTSPPTTEGFKYPRPSSVPPSPSGSQASSPQSSDVEDEVEDERYDEEEEAERDRLNIKSPFSLSHVPHGKKKLHGEYKN