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Target
Procathepsin L
Ligand
BDBM41372
Substrate
n/a
Meas. Tech.
Cathepsin L dose-response testing in the presence of cysteine
IC50
>50000±0 nM
Citation
 PubChem, PC Cathepsin L dose-response testing in the presence of cysteine PubChem Bioassay (2009)[AID] 
Target
Name:
Procathepsin L
Synonyms:
CATL1_HUMAN | CTSL | CTSL CTSL1 | CTSL1 | Cathepsin L | Cathepsin L1 | Cathepsin L1 heavy chain | Cathepsin L1 light chain | MEP | Major excreted protein | cathepsin L preproprotein
Type:
Enzyme
Mol. Mass.:
37557.19
Organism:
Homo sapiens (Human)
Description:
Purchased from Calbiochem (San Diego, CA).
Residue:
333
Sequence:
MNPTLILAAFCLGIASATLTFDHSLEAQWTKWKAMHNRLYGMNEEGWRRAVWEKNMKMIELHNQEYREGKHSFTMAMNAFGDMTSEEFRQVMNGFQNRKPRKGKVFQEPLFYEAPRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESTESDNNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV
  
Inhibitor
Name:
BDBM41372
Synonyms:
1,5-dimethyl-N-(3-morpholin-4-ylpropyl)-4-oxidanylidene-pyrrolo[3,2-c]quinoline-2-carboxamide | 1,5-dimethyl-N-(3-morpholin-4-ylpropyl)-4-oxopyrrolo[3,2-c]quinoline-2-carboxamide | 1,5-dimethyl-N-[3-(4-morpholinyl)propyl]-4-oxo-2-pyrrolo[3,2-c]quinolinecarboxamide | 4-keto-1,5-dimethyl-N-(3-morpholinopropyl)pyrrolo[3,2-c]quinoline-2-carboxamide | MLS000118084 | SMR000095032 | cid_5309031
Type:
Small organic molecule
Emp. Form.:
C21H26N4O3
Mol. Mass.:
382.4561
SMILES:
Cn1c(cc2c1c1ccccc1n(C)c2=O)C(=O)NCCCN1CCOCC1
Structure:
Search PDB for entries with ligand similarity: