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Target
Trans-activator protein BZLF1
Ligand
BDBM62469
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62469
Synonyms:
2-[(4E)-4-(3-hydroxy-4-methoxy-benzylidene)-2,5-diketo-imidazolidin-1-yl]-N-(m-tolyl)acetamide | 2-[(4E)-4-[(3-hydroxy-4-methoxyphenyl)methylidene]-2,5-dioxo-1-imidazolidinyl]-N-(3-methylphenyl)acetamide | 2-[(4E)-4-[(3-hydroxy-4-methoxyphenyl)methylidene]-2,5-dioxoimidazolidin-1-yl]-N-(3-methylphenyl)acetamide | 2-[(4E)-4-[(4-methoxy-3-oxidanyl-phenyl)methylidene]-2,5-bis(oxidanylidene)imidazolidin-1-yl]-N-(3-methylphenyl)ethanamide | 2-[4-(3-hydroxy-4-methoxybenzylidene)-2,5-dioxo-1-imidazolidinyl]-N-(3-methylphenyl)acetamide | MLS000704930 | SMR000231576 | cid_7256141
Type:
Small organic molecule
Emp. Form.:
C20H19N3O5
Mol. Mass.:
381.382
SMILES:
COc1ccc(\C=C2\NC(=O)N(CC(=O)Nc3cccc(C)c3)C2=O)cc1O
Structure:
Search PDB for entries with ligand similarity: