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Target
Oxytocin receptor
Ligand
BDBM50139178
Substrate
n/a
Meas. Tech.
ChEMBL_1681639 (CHEMBL4031916)
EC50
29±n/a nM
Citation
Lacivita, E; Perrone, R; Margari, L; Leopoldo, M Targets for Drug Therapy for Autism Spectrum Disorder: Challenges and Future Directions. J Med Chem 60:9114-9141 (2017) [PubMed] Article
More Info.:
Target
Name:
Oxytocin receptor
Synonyms:
OT-R | OXYR_MOUSE | Oxtr | Oxytocin receptor
Type:
PROTEIN
Mol. Mass.:
42826.38
Organism:
Mus musculus
Description:
ChEMBL_108294
Residue:
388
Sequence:
MEGTPAANWSIELDLGSGVPPGAEGNLTAGPPRRNEALARVEVAVLCLILFLALSGNACVLLALRTTRHKHSRLFFFMKHLSIADLVVAVFQVLPQLLWDITFRFYGPDLLCRLVKYLQVVGMFASTYLLLLMSLDRCLAICQPLRSLRRRTDRLAVLATWLGCLVASVPQVHIFSLREVADGVFDCWAVFIQPWGPKAYVTWITLAVYIVPVIVLAACYGLISFKIWQNLRLKTAAAAAAAEGSDAAGGAGRAALARVSSVKLISKAKIRTVKMTFIIVLAFIVCWTPFFFVQMWSVWDVNAPKEASAFIIAMLLASLNSCCNPWIYMLFTGHLFHELVQRFLCCSARYLKGSRPGETSISKKSNSSTFVLSRRSSSQRSCSQPSSA