Reaction Details Report a problem with these data
Target
Protein kinase domain-containing protein
Ligand
BDBM50264869
Substrate
n/a
Meas. Tech.
ChEMBL_900187 (CHEMBL3047469)
IC50
11588±n/a nM
Citation
  TBA Med Chem Res 21:681-693 (2012)    Article 
Target
Name:
Protein kinase domain-containing protein
Synonyms:
Putative uncharacterized protein pk7
Type:
PROTEIN
Mol. Mass.:
37967.83
Organism:
Plasmodium falciparum
Description:
ChEMBL_496798
Residue:
320
Sequence:
MKDILSNYSNLIYLNKYVKEKDKYINDYRIIRTLNQGKFNKIILCEKDNKFYALKKYEKSLLEKKRDFTKSNNDKISIKSKYDDFKNELQIITDIKNEYCLTCEGIITNYDEVYIIYEYMENDSILKFDEYFFVLDKNYTCFIPIQVIKCIIKSVLNSFSYIHNEKNICHRDVKPSNILMDKNGRVKLSDFGESEYMVDKKIKGSRGTYEFMPPEFFSNESSYNGAKVDIWSLGICLYVMFYNVVPFSLKISLVELFNNIRTKNIEYPLDRNHFLYPLTNKKSTCSNNFLSNEDIDFLKLFLRKNPAERITSEDALVTAK
  
Inhibitor
Name:
BDBM50264869
Synonyms:
3-(4-methoxyphenyl)-N-(pyridin-3-ylmethyl)imidazo[1,2-b]pyridazin-6-amine | CHEMBL506400
Type:
Small organic molecule
Emp. Form.:
C19H17N5O
Mol. Mass.:
331.3712
SMILES:
COc1ccc(cc1)-c1cnc2ccc(NCc3cccnc3)nn12
Structure:
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