Reaction Details Report a problem with these data
Target
Adenosine receptor A2b
Ligand
BDBM50511973
Substrate
n/a
Meas. Tech.
ChEMBL_1846291 (CHEMBL4346832)
Ki
0.234000±n/a nM
Citation
Jiang, J; Seel, CJ; Temirak, A; Namasivayam, V; Arridu, A; Schabikowski, J; Baqi, Y; Hinz, S; Hockemeyer, J; Müller, CE A J Med Chem 62:4032-4055 (2019) [PubMed] Article
More Info.:
Target
Name:
Adenosine receptor A2b
Synonyms:
AA2BR_HUMAN | ADENOSINE A2B | ADORA2B | Adenosine receptor A2B (A2B) | Adenosine receptors A2b | Adenosine receptors; A2a & A2b
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
36341.22
Organism:
Human
Description:
n/a
Residue:
332
Sequence:
MLLETQDALYVALELVIAALSVAGNVLVCAAVGTANTLQTPTNYFLVSLAAADVAVGLFAIPFAITISLGFCTDFYGCLFLACFVLVLTQSSIFSLLAVAVDRYLAICVPLRYKSLVTGTRARGVIAVLWVLAFGIGLTPFLGWNSKDSATNNCTEPWDGTTNESCCLVKCLFENVVPMSYMVYFNFFGCVLPPLLIMLVIYIKIFLVACRQLQRTELMDHSRTTLQREIHAAKSLAMIVGIFALCWLPVHAVNCVTLFQPAQGKNKPKWAMNMAILLSHANSVVNPIVYAYRNRDFRYTFHKIISRYLLCQADVKSGNGQAGVQPALGVGL