Reaction Details Report a problem with these data
Target
Retinoic acid receptor RXR-beta
Ligand
BDBM31892
Substrate
n/a
Meas. Tech.
ChEBML_197069
Kd
15±n/a nM
Citation
Farmer, LJ; Zhi, L; Jeong, S; Lamph, WW; Osburn, DL; Croston, G; Flatten, KS; Heyman, RA; Nadzan, AM Retinoic acid receptor ligands based on the 6-cyclopropyl-2,4-hexadienoic acid. Bioorg Med Chem Lett 13:261-4 (2002) [PubMed] Article
More Info.:
Target
Name:
Retinoic acid receptor RXR-beta
Synonyms:
Nr2b2 | RXRB_MOUSE | Retinoid X receptor beta | Rxrb
Type:
PROTEIN
Mol. Mass.:
55877.78
Organism:
Mouse
Description:
ChEMBL_196588
Residue:
520
Sequence:
MSWATRPPFLPPRHAAGQCGPVGVRKEMHCGVASRWRRRRPWLDPAAAAAAAGEQQALEPEPGEAGRDGMGDSGRDSRSPDSSSPNPLSQGIRPSSPPGPPLTPSAPPPPMPPPPLGSPFPVISSSMGSPGLPPPAPPGFSGPVSSPQINSTVSLPGGGSGPPEDVKPPVLGVRGLHCPPPPGGPGAGKRLCAICGDRSSGKHYGVYSCEGCKGFFKRTIRKDLTYSCRDNKDCTVDKRQRNRCQYCRYQKCLATGMKREAVQEERQRGKDKDGDGDGAGGAPEEMPVDRILEAELAVEQKSDQGVEGPGATGGGGSSPNDPVTNICQAADKQLFTLVEWAKRIPHFSSLPLDDQVILLRAGWNELLIASFSHRSIDVRDGILLATGLHVHRNSAHSAGVGAIFDRVLTELVSKMRDMRMDKTELGCLRAIILFNPDAKGLSNPGEVEILREKVYASLETYCKQKYPEQQGRFAKLLLRLPALRSIGLKCLEHLFFFKLIGDTPIDTFLMEMLEAPHQLA