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Target
Melatonin receptor type 1B
Ligand
BDBM50125649
Substrate
n/a
Meas. Tech.
ChEBML_105255
IC50
3.1±n/a nM
Citation
Mattson, RJ; Catt, JD; Keavy, D; Sloan, CP; Epperson, J; Gao, Q; Hodges, DB; Iben, L; Mahle, CD; Ryan, E; Yocca, FD Indanyl piperazines as melatonergic MT2 selective agents. Bioorg Med Chem Lett 13:1199-202 (2003) [PubMed] Article
More Info.:
Target
Name:
Melatonin receptor type 1B
Synonyms:
MTNR1B | MTR1B_HUMAN | Mel-1B-R | Mel1b melatonin receptor | Melatonin 1B | Melatonin receptor | Melatonin receptor type 1B | Melatonin receptor type 2 (MT2)
Type:
Enzyme
Mol. Mass.:
40203.54
Organism:
Human
Description:
P49286
Residue:
362
Sequence:
MSENGSFANCCEAGGWAVRPGWSGAGSARPSRTPRPPWVAPALSAVLIVTTAVDVVGNLLVILSVLRNRKLRNAGNLFLVSLALADLVVAFYPYPLILVAIFYDGWALGEEHCKASAFVMGLSVIGSVFNITAIAINRYCYICHSMAYHRIYRRWHTPLHICLIWLLTVVALLPNFFVGSLEYDPRIYSCTFIQTASTQYTAAVVVIHFLLPIAVVSFCYLRIWVLVLQARRKAKPESRLCLKPSDLRSFLTMFVVFVIFAICWAPLNCIGLAVAINPQEMAPQIPEGLFVTSYLLAYFNSCLNAIVYGLLNQNFRREYKRILLALWNPRHCIQDASKGSHAEGLQSPAPPIIGVQHQADAL